| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4854493 | 14 | PB | = | 98.4 | % | ALA4836426 | % | ||||
| 2. | ALA4854493 | 14 | F | = | 25 | % | ALA4836425 | % | ||||
| 3. | ALA4854493 | 14 | t1/2 | = | 6.2 | hr | ALA4836424 | hr | ||||
| 4. | ALA4854493 | 14 | CL | = | 8 | ml/min.kg | ALA4836423 | mL.min-1.kg-1 | ||||
| 5. | ALA4854493 | 14 | INH | = | 45 | % | ALA4836419 | % | Mus musculus | |||
| 6. | ALA4854493 | 14 | FC | > | 10 | ALA4836418 | Mus musculus | |||||
| 7. | ALA4854493 | 14 | Activity | 0 | ALA4836417 | Not Active | Mus musculus | |||||
| 8. | ALA4854493 | 14 | Ratio | = | 0.43 | ALA4836416 | ||||||
| 9. | ALA4854493 | 14 | Drug uptake | = | 629 | ng/g | ALA4836415 | ng/g | ||||
| 10. | ALA4854493 | 14 | Cp | = | 1402 | ng/ml | ALA4836414 | ng/ml | ||||
| 11. | ALA4854493 | 14 | Drug metabolism | = | 0.092 | umol/ml | ALA4836405 | umol/ml | ||||
| 12. | ALA4854493 | 14 | CLH | = | 0.218 | uL/min | ALA4836404 | uL/min | ||||
| 13. | ALA4854493 | 14 | CLH | = | 0.068 | uL/min | ALA4836403 | uL/min | ||||
| 14. | ALA4854493 | 14 | IC50 | = | 12.8 | nM | ALA4836402 | 7.89 | nM | Homo sapiens |
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