# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4856135 | 49; HSD1237 | INH | = | 90 | % | ALA4836811 | % | Homo sapiens | |||
2. | ALA4856135 | 49; HSD1237 | Activity | 0 | ALA4836810 | Active | Homo sapiens | |||||
3. | ALA4856135 | 49; HSD1237 | Activity | 0 | ALA4836809 | Active | Homo sapiens | |||||
4. | ALA4856135 | 49; HSD1237 | Activity | 0 | ALA4836808 | Active | Homo sapiens | |||||
5. | ALA4856135 | 49; HSD1237 | Activity | 0 | ALA4836807 | Active | Homo sapiens | |||||
6. | ALA4856135 | 49; HSD1237 | Activity | 0 | ALA4836806 | Active | Homo sapiens | |||||
7. | ALA4856135 | 49; HSD1237 | INH | 0 | ALA4836805 | Not Active | % | Homo sapiens | ||||
8. | ALA4856135 | 49; HSD1237 | INH | 0 | ALA4836804 | Active | % | Homo sapiens | ||||
9. | ALA4856135 | 49; HSD1237 | INH | 0 | ALA4836803 | Active | % | Homo sapiens | ||||
10. | ALA4856135 | 49; HSD1237 | Kd | = | 1.3 | nM | ALA4836802 | 8.89 | nM | Homo sapiens | ||
11. | ALA4856135 | 49; HSD1237 | Kd | = | 0.73 | nM | ALA4836801 | 9.14 | nM | Homo sapiens | ||
12. | ALA4856135 | 49; HSD1237 | Kd | = | 1.6 | nM | ALA4836800 | 8.80 | nM | Homo sapiens | ||
13. | ALA4856135 | 49; HSD1237 | Activity | = | 4 | % | ALA4836792 | % | Homo sapiens | |||
14. | ALA4856135 | 49; HSD1237 | Activity | = | 4 | % | ALA4836791 | % | Homo sapiens | |||
15. | ALA4856135 | 49; HSD1237 | Activity | = | 4 | % | ALA4836790 | % | Homo sapiens | |||
16. | ALA4856135 | 49; HSD1237 | Activity | = | 4 | % | ALA4836789 | % | Homo sapiens | |||
17. | ALA4856135 | 49; HSD1237 | Activity | = | 4 | % | ALA4836788 | % | Homo sapiens | |||
18. | ALA4856135 | 49; HSD1237 | Activity | < | 2.5 | % | ALA4836787 | % | Homo sapiens | |||
19. | ALA4856135 | 49; HSD1237 | Activity | < | 2.5 | % | ALA4836786 | % | Homo sapiens | |||
20. | ALA4856135 | 49; HSD1237 | IC50 | = | 0.062 | uM | ALA4836785 | 7.21 | nM | Mus musculus |