# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4856311 | 24 | Stability | 0 | ALA4841991 | Stable | % | |||||
2. | ALA4856311 | 24 | t1/2 | = | 2.6 | hr | ALA4841990 | hr | ||||
3. | ALA4856311 | 24 | Stability | 0 | ALA4841989 | Not Determined | % | |||||
4. | ALA4856311 | 24 | Stability | = | 19 | % | ALA4841988 | % | ||||
5. | ALA4856311 | 24 | Stability | = | 57 | % | ALA4841987 | % | ||||
6. | ALA4856311 | 24 | Stability | = | 87 | % | ALA4841986 | % | ||||
7. | ALA4856311 | 24 | Stability | = | 94 | % | ALA4841985 | % | ||||
8. | ALA4856311 | 24 | Stability | 0 | ALA4841984 | Stable | % | |||||
9. | ALA4856311 | 24 | Intrinsic activity | = | 0.95 | % | ALA4841983 | % | Homo sapiens | |||
10. | ALA4856311 | 24 | pEC50 | = | 8.85 | ALA4841982 | 8.85 | nM | Homo sapiens | |||
11. | ALA4856311 | 24 | Intrinsic activity | = | 0.84 | % | ALA4841981 | % | Homo sapiens | |||
12. | ALA4856311 | 24 | pEC50 | = | 9 | ALA4841980 | 9.00 | nM | Homo sapiens | |||
13. | ALA4856311 | 24 | Intrinsic activity | = | 0.8 | % | ALA4841979 | % | Homo sapiens | |||
14. | ALA4856311 | 24 | pEC50 | = | 8.78 | ALA4841978 | 8.78 | nM | Homo sapiens | |||
15. | ALA4856311 | 24 | Intrinsic activity | = | 0.98 | % | ALA4841977 | % | Homo sapiens | |||
16. | ALA4856311 | 24 | EC50 | = | 1 | nM | ALA4841976 | 9.00 | nM | Homo sapiens | ||
17. | ALA4856311 | 24 | pEC50 | = | 9 | ALA4841976 | 9.00 | nM | Homo sapiens | |||
18. | ALA4856311 | 24 | Selectivity ratio | > | 90000 | ALA4841975 | ||||||
19. | ALA4856311 | 24 | Selectivity ratio | > | 300 | ALA4841974 | ||||||
20. | ALA4856311 | 24 | Selectivity ratio | > | 300000 | ALA4841973 |