# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4856716 | 2 | INH | = | 55 | % | ALA4806279 | % | Homo sapiens | |||
2. | ALA4856716 | 2 | INH | = | 2 | % | ALA4806278 | % | Homo sapiens | |||
3. | ALA4856716 | 2 | INH | = | 23 | % | ALA4806277 | % | Homo sapiens | |||
4. | ALA4856716 | 2 | INH | = | 5 | % | ALA4806276 | % | Homo sapiens | |||
5. | ALA4856716 | 2 | t1/2 | = | 18 | min | ALA4806275 | hr | ||||
6. | ALA4856716 | 2 | t1/2 | = | 11 | min | ALA4806274 | hr | ||||
7. | ALA4856716 | 2 | t1/2 | = | 39 | min | ALA4806273 | hr | ||||
8. | ALA4856716 | 2 | solubility | = | 0.8 | uM | ALA4806272 | nM | ||||
9. | ALA4856716 | 2 | GI50 | = | 66 | nM | ALA4806271 | nM | Homo sapiens | |||
10. | ALA4856716 | 2 | GI50 | = | 95 | nM | ALA4806270 | nM | Homo sapiens | |||
11. | ALA4856716 | 2 | IC50 | = | 2200 | nM | ALA4806269 | 5.66 | nM | |||
12. | ALA4856716 | 2 | IC50 | = | 6500 | nM | ALA4806266 | 5.19 | nM | Homo sapiens | ||
13. | ALA4856716 | 2 | IC50 | > | 9900 | nM | ALA4806265 | nM | Homo sapiens |