| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4857486 | 2a | INH | 0 | ALA4832695 | Not Active | % | |||||
| 2. | ALA4857486 | 2a | INH | = | 11 | % | ALA4832694 | % | ||||
| 3. | ALA4857486 | 2a | INH | = | 22 | % | ALA4832693 | % | ||||
| 4. | ALA4857486 | 2a | INH | 0 | ALA4832692 | Not Active | % | Homo sapiens | ||||
| 5. | ALA4857486 | 2a | CC50 | > | 100 | uM | ALA4832691 | nM | Homo sapiens | |||
| 6. | ALA4857486 | 2a | CC50 | 0 | ALA4832690 | Not Determined | Mus musculus | |||||
| 7. | ALA4857486 | 2a | EC50 | = | 4.8 | uM | ALA4832688 | 5.32 | nM | Trypanosoma brucei brucei | ||
| 8. | ALA4857486 | 2a | Activity | 0 | ALA4832687 | Active | Trypanosoma brucei rhodesiense | |||||
| 9. | ALA4857486 | 2a | K | = | 0.01 | /s | ALA4832684 | /s | Trypanosoma brucei rhodesiense | |||
| 10. | ALA4857486 | 2a | K | = | 0.055 | /s | ALA4832683 | /s | Trypanosoma brucei rhodesiense | |||
| 11. | ALA4857486 | 2a | Selectivity Index | = | 4 | ALA4832679 | ||||||
| 12. | ALA4857486 | 2a | Ki | = | 1.7 | uM | ALA4832678 | 5.77 | nM | Homo sapiens | ||
| 13. | ALA4857486 | 2a | Ki | = | 0.06 | uM | ALA4832677 | 7.22 | nM | Homo sapiens | ||
| 14. | ALA4857486 | 2a | Ki | = | 0.258 | uM | ALA4832676 | 6.59 | nM | Homo sapiens | ||
| 15. | ALA4857486 | 2a | Ki | = | 0.015 | uM | ALA4832675 | 7.82 | nM | Trypanosoma brucei rhodesiense | ||
| 16. | ALA4857486 | 2a | Ki | = | 0.098 | uM | ALA4832674 | 7.01 | nM | Trypanosoma brucei rhodesiense |
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