| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4857808 | 12 | Activity | 0 | ALA4834341 | Non-Toxic | ||||||
| 2. | ALA4857808 | 12 | Activity | 0 | ALA4834340 | Active | Mus musculus | |||||
| 3. | ALA4857808 | 12 | Activity | 0 | ALA4834339 | Non-Toxic | ||||||
| 4. | ALA4857808 | 12 | fCmax | = | 0.031 | uM | ALA4834331 | uM | ||||
| 5. | ALA4857808 | 12 | fAUC | = | 0.45 | uM.hr | ALA4834328 | uM.hr | ||||
| 6. | ALA4857808 | 12 | Cmax | = | 7.4 | uM | ALA4834325 | nM | ||||
| 7. | ALA4857808 | 12 | AUC | = | 106 | uM.hr | ALA4834322 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 8. | ALA4857808 | 12 | PPB | = | 99.58 | % | ALA4834319 | % | ||||
| 9. | ALA4857808 | 12 | IC50 | = | 3 | uM | ALA4834318 | 5.52 | nM | Homo sapiens | ||
| 10. | ALA4857808 | 12 | IC50 | = | 9.9 | uM | ALA4834317 | 5.00 | nM | Homo sapiens | ||
| 11. | ALA4857808 | 12 | IC50 | = | 0.11 | uM | ALA4834316 | 6.96 | nM | Homo sapiens | ||
| 12. | ALA4857808 | 12 | Ratio | = | 0.34 | ALA4834315 | ||||||
| 13. | ALA4857808 | 12 | Ratio | = | 0.4 | ALA4834314 | ||||||
| 14. | ALA4857808 | 12 | F | = | 58 | % | ALA4834313 | % | ||||
| 15. | ALA4857808 | 12 | Cmax | = | 9.5 | uM | ALA4834311 | nM | ||||
| 16. | ALA4857808 | 12 | Cmax | = | 5.6 | uM | ALA4834310 | nM | ||||
| 17. | ALA4857808 | 12 | AUC | = | 160 | uM.hr | ALA4834307 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 18. | ALA4857808 | 12 | AUC | = | 54 | uM.hr | ALA4834306 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 19. | ALA4857808 | 12 | t1/2 | = | 22 | hr | ALA4834303 | hr | ||||
| 20. | ALA4857808 | 12 | t1/2 | = | 10 | hr | ALA4834302 | hr |
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