| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4858136 | 31 | IC50 | = | 6.8 | uM | ALA4845530 | 5.17 | nM | Homo sapiens | ||
| 2. | ALA4858136 | 31 | Activity | 0 | ALA4845529 | Not Active | Homo sapiens | |||||
| 3. | ALA4858136 | 31 | Activity | 0 | ALA4845528 | Not Active | Homo sapiens | |||||
| 4. | ALA4858136 | 31 | Activity | 0 | ALA4845527 | Not Active | Homo sapiens | |||||
| 5. | ALA4858136 | 31 | Activity | 0 | ALA4845526 | Not Active | Homo sapiens | |||||
| 6. | ALA4858136 | 31 | Activity | 0 | ALA4845525 | Not Active | Homo sapiens | |||||
| 7. | ALA4858136 | 31 | Activity | 0 | ALA4845524 | Not Active | Homo sapiens | |||||
| 8. | ALA4858136 | 31 | Activity | 0 | ALA4845523 | Not Active | Homo sapiens | |||||
| 9. | ALA4858136 | 31 | F | = | 24 | % | ALA4845522 | % | ||||
| 10. | ALA4858136 | 31 | t1/2 | = | 3.5 | hr | ALA4845521 | hr | ||||
| 11. | ALA4858136 | 31 | AUC | = | 4001 | hr.ng/ml | ALA4845520 | ng.hr.mL-1 | ||||
| 12. | ALA4858136 | 31 | Vd | = | 9.35 | L/Kg | ALA4845517 | L.kg-1 | ||||
| 13. | ALA4858136 | 31 | CL | = | 1.83 | L/hr/kg | ALA4845516 | mL.min-1.kg-1 | ||||
| 14. | ALA4858136 | 31 | Cmax | = | 297 | ng/ml | ALA4845515 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 15. | ALA4858136 | 31 | Cmax | = | 791 | ng/ml | ALA4845514 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 16. | ALA4858136 | 31 | IC50 | > | 20 | uM | ALA4845512 | nM | Homo sapiens | |||
| 17. | ALA4858136 | 31 | permeability | = | 235 | nm/s | ALA4845511 | nm/s | ||||
| 18. | ALA4858136 | 31 | IC50 | > | 20 | uM | ALA4845510 | nM | Homo sapiens | |||
| 19. | ALA4858136 | 31 | Stabilty | = | 85.8 | % | ALA4845509 | % | ||||
| 20. | ALA4858136 | 31 | Stabilty | = | 21 | % | ALA4845508 | % |
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