Activities

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Activities

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#	Name	Compound Key	Action Type	Relation	Activity Value	Units	Assay ID	Assay Description	Comment	Assay	Assay Organism
1.	ALA4858811	5; JNJ-63576253	TGI	=	87	%	ALA5140978			%	Homo sapiens
2.	ALA4858811	5; JNJ-63576253	F	=	45	%	ALA5140977			%
3.	ALA4858811	5; JNJ-63576253	IC50	=	290	nM	ALA5140976	6.54		nM	Homo sapiens
4.	ALA4858811	5; JNJ-63576253	IC50	=	37	nM	ALA5140975	7.43		nM	Homo sapiens
5.	ALA4858811	5; JNJ-63576253	IC50	=	54	nM	ALA5140974	7.27		nM	Homo sapiens
6.	ALA4858811	5; JNJ-63576253	F	=	45	%	ALA4820525			%
7.	ALA4858811	5; JNJ-63576253	Vdss	=	6.11	L/Kg	ALA4820524			L.kg-1
8.	ALA4858811	5; JNJ-63576253	t1/2	=	5.99	hr	ALA4820523			hr
9.	ALA4858811	5; JNJ-63576253	CL	=	15	ml/min.kg	ALA4820522			mL.min-1.kg-1
10.	ALA4858811	5; JNJ-63576253	Cmax	=	0.66	uM	ALA4820521			nM
11.	ALA4858811	5; JNJ-63576253	AUClast	=	4.9	microg.hr/mL	ALA4820520			ng.hr.mL-1
12.	ALA4858811	5; JNJ-63576253	Papp	=	5.62	10^-6 cm/s	ALA4820519			10^-6 cm/s
13.	ALA4858811	5; JNJ-63576253	t1/2	>	180	min	ALA4820518			hr
14.	ALA4858811	5; JNJ-63576253	Drug metabolism	=	0.6	%	ALA4820517			%
15.	ALA4858811	5; JNJ-63576253	Drug metabolism	=	0.6	%	ALA4820516			%
16.	ALA4858811	5; JNJ-63576253	Drug metabolism	=	0.6	%	ALA4820514			%
17.	ALA4858811	5; JNJ-63576253	Drug metabolism	=	98.8	%	ALA4820513			%
18.	ALA4858811	5; JNJ-63576253	Drug metabolism	=	100	%	ALA4820512			%
19.	ALA4858811	5; JNJ-63576253	Ct	=	1750	ng/ml	ALA4820497			ng/ml
20.	ALA4858811	5; JNJ-63576253	INH		0		ALA4820496		Active	%	Rattus norvegicus