# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4859105 | 27; BRD0639 | IC50 | = | 568 | nM | ALA5218139 | 6.25 | nM | |||
2. | ALA4859105 | 27; BRD0639 | Activity | 0 | ALA4827812 | Active | Homo sapiens | |||||
3. | ALA4859105 | 27; BRD0639 | IC50 | = | 16 | uM | ALA4827811 | 4.80 | nM | |||
4. | ALA4859105 | 27; BRD0639 | IC50 | = | 7.5 | uM | ALA4827810 | 5.12 | nM | Homo sapiens | ||
5. | ALA4859105 | 27; BRD0639 | EC50 | = | 3 | uM | ALA4827809 | 5.52 | nM | Homo sapiens | ||
6. | ALA4859105 | 27; BRD0639 | Ratio | = | 244 | /M/s | ALA4827808 | /M/s | Homo sapiens | |||
7. | ALA4859105 | 27; BRD0639 | Ki | = | 49 | uM | ALA4827807 | 4.31 | nM | Homo sapiens | ||
8. | ALA4859105 | 27; BRD0639 | Kinact | = | 0.715 | /min | ALA4827806 | /min | Homo sapiens | |||
9. | ALA4859105 | 27; BRD0639 | t1/2 | = | 916 | min | ALA4827799 | hr | ||||
10. | ALA4859105 | 27; BRD0639 | Stabilty | = | 79 | % | ALA4827798 | % | ||||
11. | ALA4859105 | 27; BRD0639 | Stabilty | = | 87 | % | ALA4827797 | % | ||||
12. | ALA4859105 | 27; BRD0639 | solubility | = | 82 | uM | ALA4827796 | nM | ||||
13. | ALA4859105 | 27; BRD0639 | IC50 | = | 13.8 | uM | ALA4827795 | 4.86 | nM | Homo sapiens |