# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4859858 | 7 | ED50 | > | 100 | mg kg-1 | ALA5236049 | mg.kg-1 | Mus musculus | |||
2. | ALA4859858 | 7 | Activity | 0 | ALA5236046 | Not Active | Mus musculus | |||||
3. | ALA4859858 | 7 | Emax | = | 43 | % | ALA5236042 | % | Mus musculus | |||
4. | ALA4859858 | 7 | EC50 | = | 6225.7 | nM | ALA5236041 | 5.21 | nM | Mus musculus | ||
5. | ALA4859858 | 7 | Ki | = | 7947 | nM | ALA5236040 | 5.10 | nM | Mus musculus | ||
6. | ALA4859858 | 7 | Ki | = | 2198 | nM | ALA5236039 | 5.66 | nM | Mus musculus | ||
7. | ALA4859858 | 7 | Ki | = | 578.23 | nM | ALA5236038 | 6.24 | nM | Mus musculus | ||
8. | ALA4859858 | 7 | IC50 | = | 10000 | nM | ALA5127645 | 5.00 | nM | Homo sapiens | ||
9. | ALA4859858 | 7 | IC50 | > | 10000 | nM | ALA5127644 | nM | Homo sapiens | |||
10. | ALA4859858 | 7 | IC50 | = | 5700 | nM | ALA5127643 | 5.24 | nM | Homo sapiens | ||
11. | ALA4859858 | 7 | Ki | = | 3200 | nM | ALA5127527 | 5.50 | nM | Homo sapiens | ||
12. | ALA4859858 | 7 | Ki | > | 10000 | nM | ALA5127526 | nM | Homo sapiens | |||
13. | ALA4859858 | 7 | Ki | = | 728 | nM | ALA5127525 | 6.14 | nM | Homo sapiens | ||
14. | ALA4859858 | 7 | Ki | = | 728 | nM | ALA4808365 | 6.14 | nM | Homo sapiens | ||
15. | ALA4859858 | 7 | Drug recovery | > | 80 | % | ALA4834835 | % | ||||
16. | ALA4859858 | 7 | Drug recovery | > | 90 | % | ALA4834834 | % | ||||
17. | ALA4859858 | 7 | Cp | < | 1 | ng/ml | ALA4834827 | ng/ml | ||||
18. | ALA4859858 | 7 | Cp | < | 1 | ng/ml | ALA4834826 | ng/ml | ||||
19. | ALA4859858 | 7 | Cmax | = | 2.9 | ng/ml | ALA4834821 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
20. | ALA4859858 | 7 | Tmax | = | 5 | min | ALA4834820 | hr |