| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4859955 | DB1263 | Time | = | 22.75 | day | ALA4827168 | hr | Trypanosoma brucei rhodesiense | |||
| 2. | ALA4859955 | DB1263 | Selectivity Index | = | 64.5 | ALA4827167 | ||||||
| 3. | ALA4859955 | DB1263 | Selectivity Index | = | 57.1 | ALA4827166 | ||||||
| 4. | ALA4859955 | DB1263 | IC50 | = | 31 | nM | ALA4827165 | 7.51 | nM | Plasmodium falciparum | ||
| 5. | ALA4859955 | DB1263 | IC50 | = | 35 | nM | ALA4827164 | 7.46 | nM | Trypanosoma brucei rhodesiense | ||
| 6. | ALA4859955 | DB1263 | deltaTm | = | 8.5 | degrees C | ALA4827163 | degrees C | ||||
| 7. | ALA4859955 | DB1263 | IC50 | = | 2 | uM | ALA4827162 | 5.70 | nM | Rattus norvegicus | ||
| 8. | ALA4859955 | DB1263 | Activity | > | 50 | % | ALA4814083 | % | Homo sapiens |
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