# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4860336 | 2b | MRT | = | 1.57 | hr | ALA4831402 | hr | ||||
2. | ALA4860336 | 2b | AUC | = | 168 | hr.ng/ml | ALA4831401 | ng.hr.mL-1 | ||||
3. | ALA4860336 | 2b | AUCt | = | 166 | hr.ng/ml | ALA4831400 | ng.hr.mL-1 | ||||
4. | ALA4860336 | 2b | Cmax | = | 127 | ng/ml | ALA4831399 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
5. | ALA4860336 | 2b | Tmax | = | 1.08 | hr | ALA4831398 | hr | ||||
6. | ALA4860336 | 2b | t1/2 | = | 0.7 | hr | ALA4831397 | hr | ||||
7. | ALA4860336 | 2b | INH | = | 91.6 | % | ALA4831396 | % | Homo sapiens | |||
8. | ALA4860336 | 2b | IC50 | = | 1.39 | uM | ALA4831395 | 5.86 | nM | Homo sapiens | ||
9. | ALA4860336 | 2b | IC50 | = | 0.33 | uM | ALA4831394 | 6.48 | nM | Homo sapiens | ||
10. | ALA4860336 | 2b | IC50 | = | 7.6 | nM | ALA4831392 | 8.12 | nM | Homo sapiens |