# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4860770 | 2e | INH | = | 11 | % | ALA4832695 | % | ||||
2. | ALA4860770 | 2e | INH | = | 22 | % | ALA4832694 | % | ||||
3. | ALA4860770 | 2e | INH | = | 31 | % | ALA4832693 | % | ||||
4. | ALA4860770 | 2e | INH | 0 | ALA4832692 | Not Active | % | Homo sapiens | ||||
5. | ALA4860770 | 2e | CC50 | > | 100 | uM | ALA4832691 | nM | Homo sapiens | |||
6. | ALA4860770 | 2e | CC50 | 0 | ALA4832690 | Not Determined | Mus musculus | |||||
7. | ALA4860770 | 2e | EC50 | = | 0.14 | uM | ALA4832688 | 6.85 | nM | Trypanosoma brucei brucei | ||
8. | ALA4860770 | 2e | K | = | 0.005 | /s | ALA4832684 | /s | Trypanosoma brucei rhodesiense | |||
9. | ALA4860770 | 2e | K | = | 0.065 | /s | ALA4832683 | /s | Trypanosoma brucei rhodesiense | |||
10. | ALA4860770 | 2e | INH | = | 14 | % | ALA4832680 | % | Homo sapiens | |||
11. | ALA4860770 | 2e | Selectivity Index | = | 6 | ALA4832679 | ||||||
12. | ALA4860770 | 2e | Ki | = | 0.039 | uM | ALA4832677 | 7.41 | nM | Homo sapiens | ||
13. | ALA4860770 | 2e | Ki | = | 0.348 | uM | ALA4832676 | 6.46 | nM | Homo sapiens | ||
14. | ALA4860770 | 2e | Ki | = | 0.007 | uM | ALA4832675 | 8.15 | nM | Trypanosoma brucei rhodesiense | ||
15. | ALA4860770 | 2e | Ki | = | 0.098 | uM | ALA4832674 | 7.01 | nM | Trypanosoma brucei rhodesiense |