# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4861217 | 11 | Activity | = | 2 | % | ALA4836691 | % | ||||
2. | ALA4861217 | 11 | Activity | = | 68 | % | ALA4836686 | % | Homo sapiens | |||
3. | ALA4861217 | 11 | PPB | = | 84 | % | ALA4836680 | % | ||||
4. | ALA4861217 | 11 | PPB | = | 92.6 | % | ALA4836679 | % | ||||
5. | ALA4861217 | 11 | F | = | 20 | % | ALA4836678 | % | ||||
6. | ALA4861217 | 11 | AUC | = | 0.16 | ug.hr/ml | ALA4836677 | ng.hr.mL-1 | ||||
7. | ALA4861217 | 11 | Vdss | = | 4.7 | L/Kg | ALA4836676 | L.kg-1 | ||||
8. | ALA4861217 | 11 | CL | = | 1.3 | ml/hr.kg | ALA4836675 | mL.min-1.kg-1 | ||||
9. | ALA4861217 | 11 | t1/2 | = | 3.2 | hr | ALA4836674 | hr | ||||
10. | ALA4861217 | 11 | IC50 | = | 0.21 | uM | ALA4836673 | 6.68 | nM | Homo sapiens | ||
11. | ALA4861217 | 11 | IC50 | = | 0.097 | uM | ALA4836672 | 7.01 | nM | Homo sapiens | ||
12. | ALA4861217 | 11 | IC50 | = | 0.064 | uM | ALA4836671 | 7.19 | nM | Homo sapiens |