# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4861941 | 2d | INH | 0 | ALA4832695 | Not Active | % | |||||
2. | ALA4861941 | 2d | INH | = | 20 | % | ALA4832694 | % | ||||
3. | ALA4861941 | 2d | INH | = | 44 | % | ALA4832693 | % | ||||
4. | ALA4861941 | 2d | INH | = | 10 | % | ALA4832692 | % | Homo sapiens | |||
5. | ALA4861941 | 2d | CC50 | > | 100 | uM | ALA4832691 | nM | Homo sapiens | |||
6. | ALA4861941 | 2d | CC50 | 0 | ALA4832690 | Not Determined | Mus musculus | |||||
7. | ALA4861941 | 2d | EC50 | = | 1.9 | uM | ALA4832689 | 5.72 | nM | Trypanosoma brucei brucei | ||
8. | ALA4861941 | 2d | Activity | = | 89 | % | ALA4832686 | % | Trypanosoma brucei rhodesiense | |||
9. | ALA4861941 | 2d | K | = | 0.01 | /s | ALA4832684 | /s | Trypanosoma brucei rhodesiense | |||
10. | ALA4861941 | 2d | K | = | 0.075 | /s | ALA4832683 | /s | Trypanosoma brucei rhodesiense | |||
11. | ALA4861941 | 2d | INH | = | 38 | % | ALA4832680 | % | Homo sapiens | |||
12. | ALA4861941 | 2d | Selectivity Index | = | 26 | ALA4832679 | ||||||
13. | ALA4861941 | 2d | Ki | = | 0.078 | uM | ALA4832677 | 7.11 | nM | Homo sapiens | ||
14. | ALA4861941 | 2d | Ki | = | 0.313 | uM | ALA4832676 | 6.50 | nM | Homo sapiens | ||
15. | ALA4861941 | 2d | Ki | = | 0.003 | uM | ALA4832675 | 8.52 | nM | Trypanosoma brucei rhodesiense | ||
16. | ALA4861941 | 2d | Ki | = | 0.024 | uM | ALA4832674 | 7.62 | nM | Trypanosoma brucei rhodesiense |