| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4862140 | 21 | Intrinsic activity | 0 | ALA4841981 | Not Determined | Homo sapiens | |||||
| 2. | ALA4862140 | 21 | pEC50 | 0 | ALA4841980 | Not Determined | Homo sapiens | |||||
| 3. | ALA4862140 | 21 | Intrinsic activity | = | 0.61 | % | ALA4841979 | % | Homo sapiens | |||
| 4. | ALA4862140 | 21 | pEC50 | = | 6.53 | ALA4841978 | 6.53 | nM | Homo sapiens | |||
| 5. | ALA4862140 | 21 | Intrinsic activity | = | 0.57 | % | ALA4841977 | % | Homo sapiens | |||
| 6. | ALA4862140 | 21 | EC50 | = | 270 | nM | ALA4841976 | 6.57 | nM | Homo sapiens | ||
| 7. | ALA4862140 | 21 | pEC50 | = | 6.57 | ALA4841976 | 6.57 | nM | Homo sapiens | |||
| 8. | ALA4862140 | 21 | Selectivity ratio | > | 1000 | ALA4841975 | ||||||
| 9. | ALA4862140 | 21 | Selectivity ratio | > | 1400 | ALA4841974 | ||||||
| 10. | ALA4862140 | 21 | Selectivity ratio | > | 1400 | ALA4841973 | ||||||
| 11. | ALA4862140 | 21 | Ki | > | 10000 | nM | ALA4841972 | nM | Homo sapiens | |||
| 12. | ALA4862140 | 21 | pKi | < | 5 | ALA4841972 | nM | Homo sapiens | ||||
| 13. | ALA4862140 | 21 | Ki | > | 10000 | nM | ALA4841971 | nM | Homo sapiens | |||
| 14. | ALA4862140 | 21 | pKi | < | 5 | ALA4841971 | nM | Homo sapiens | ||||
| 15. | ALA4862140 | 21 | Ki | > | 10000 | nM | ALA4841970 | nM | Homo sapiens | |||
| 16. | ALA4862140 | 21 | pKi | < | 5 | ALA4841970 | nM | Homo sapiens | ||||
| 17. | ALA4862140 | 21 | FC | = | -2.1 | ALA4841969 | Homo sapiens | |||||
| 18. | ALA4862140 | 21 | Ki | = | 7.1 | nM | ALA4841968 | 8.15 | nM | Homo sapiens | ||
| 19. | ALA4862140 | 21 | pKi | = | 8.16 | ALA4841968 | 8.16 | nM | Homo sapiens |
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