# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4863549 | A23 | INH | > | 45 | % | ALA4835403 | % | Homo sapiens | |||
2. | ALA4863549 | A23 | Activity | 0 | ALA4835402 | Not Active | Mus musculus | |||||
3. | ALA4863549 | A23 | Activity | 0 | ALA4835401 | Not Active | Mus musculus | |||||
4. | ALA4863549 | A23 | Activity | = | 1.8 | ALA4835400 | Mus musculus | |||||
5. | ALA4863549 | A23 | Activity | = | 39.8 | % | ALA4835399 | % | Mus musculus | |||
6. | ALA4863549 | A23 | Activity | = | 38.5 | % | ALA4835398 | % | Mus musculus | |||
7. | ALA4863549 | A23 | Activity | = | 38.9 | % | ALA4835397 | % | Mus musculus | |||
8. | ALA4863549 | A23 | F | = | 84.8 | % | ALA4835396 | % | ||||
9. | ALA4863549 | A23 | F | = | 90.4 | % | ALA4835395 | % | ||||
10. | ALA4863549 | A23 | MRT | = | 2.25 | hr | ALA4835394 | hr | ||||
11. | ALA4863549 | A23 | MRT | = | 1.7 | hr | ALA4835393 | hr | ||||
12. | ALA4863549 | A23 | MRT | = | 1.19 | hr | ALA4835392 | hr | ||||
13. | ALA4863549 | A23 | CL | = | 62.5 | ml/hr.kg | ALA4835391 | mL.min-1.kg-1 | ||||
14. | ALA4863549 | A23 | CL | = | 52.9 | ml/hr.kg | ALA4835390 | mL.min-1.kg-1 | ||||
15. | ALA4863549 | A23 | CL | = | 55 | ml/hr.kg | ALA4835389 | mL.min-1.kg-1 | ||||
16. | ALA4863549 | A23 | AUC | = | 160.13 | hr.microg/ml | ALA4835388 | ng.hr.mL-1 | ||||
17. | ALA4863549 | A23 | AUC | = | 18.89 | hr.microg/ml | ALA4835387 | ng.hr.mL-1 | ||||
18. | ALA4863549 | A23 | AUC | = | 5.45 | hr.microg/ml | ALA4835386 | ng.hr.mL-1 | ||||
19. | ALA4863549 | A23 | AUCt | = | 156.63 | hr.microg/ml | ALA4835385 | ng.hr.mL-1 | ||||
20. | ALA4863549 | A23 | AUCt | = | 18.46 | hr.microg/ml | ALA4835384 | ng.hr.mL-1 |