# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4864352 | S2157 | Ki | > | 250 | uM | ALA4814431 | nM | Homo sapiens | |||
2. | ALA4864352 | S2157 | Ki | > | 250 | uM | ALA4814430 | nM | Homo sapiens | |||
3. | ALA4864352 | S2157 | Ki | > | 250 | uM | ALA4814429 | nM | Homo sapiens | |||
4. | ALA4864352 | S2157 | Ki | = | 0.37 | uM | ALA4814428 | 6.43 | nM | Homo sapiens | ||
5. | ALA4864352 | S2157 | INH | 0 | ALA5135958 | Active | % | Homo sapiens | ||||
6. | ALA4864352 | S2157 | t1/2 | = | 0.95 | hr | ALA5135957 | hr | ||||
7. | ALA4864352 | S2157 | Tmax | = | 0.25 | hr | ALA5135956 | hr | ||||
8. | ALA4864352 | S2157 | Cmax | = | 0.96 | uM | ALA5135955 | nM | ||||
9. | ALA4864352 | S2157 | AUC | = | 0.98 | uM.hr | ALA5135954 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
10. | ALA4864352 | S2157 | INH | = | 51 | % | ALA5135948 | % | Homo sapiens | |||
11. | ALA4864352 | S2157 | Ratio | = | 6000 | /M/s | ALA5135947 | /M/s | Homo sapiens | |||
12. | ALA4864352 | S2157 | Ki | = | 0.75 | uM | ALA5135946 | 6.12 | nM | Homo sapiens | ||
13. | ALA4864352 | S2157 | Kinact | = | 0.005 | 10^-4/s | ALA5135945 | 10^-4/s | Homo sapiens | |||
14. | ALA4864352 | S2157 | IC50 | = | 0.87 | uM | ALA5135944 | 6.06 | nM | Homo sapiens | ||
15. | ALA4864352 | S2157 | IC50 | > | 50 | uM | ALA5053594 | nM | Homo sapiens |