| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4865048 | 17 | Stability | 0 | ALA4841991 | Stable | % | |||||
| 2. | ALA4865048 | 17 | t1/2 | = | 5.9 | hr | ALA4841990 | hr | ||||
| 3. | ALA4865048 | 17 | Stability | = | 3 | % | ALA4841989 | % | ||||
| 4. | ALA4865048 | 17 | Stability | = | 49 | % | ALA4841988 | % | ||||
| 5. | ALA4865048 | 17 | Stability | = | 91 | % | ALA4841987 | % | ||||
| 6. | ALA4865048 | 17 | Stability | 0 | ALA4841986 | Not Determined | % | |||||
| 7. | ALA4865048 | 17 | Stability | > | 99 | % | ALA4841985 | % | ||||
| 8. | ALA4865048 | 17 | Intrinsic activity | = | 0.88 | % | ALA4841983 | % | Homo sapiens | |||
| 9. | ALA4865048 | 17 | pEC50 | = | 7.77 | ALA4841982 | 7.77 | nM | Homo sapiens | |||
| 10. | ALA4865048 | 17 | Intrinsic activity | = | 0.7 | % | ALA4841981 | % | Homo sapiens | |||
| 11. | ALA4865048 | 17 | pEC50 | = | 6.69 | ALA4841980 | 6.69 | nM | Homo sapiens | |||
| 12. | ALA4865048 | 17 | Intrinsic activity | = | 0.83 | % | ALA4841979 | % | Homo sapiens | |||
| 13. | ALA4865048 | 17 | pEC50 | = | 6.85 | ALA4841978 | 6.85 | nM | Homo sapiens | |||
| 14. | ALA4865048 | 17 | Intrinsic activity | = | 0.75 | % | ALA4841977 | % | Homo sapiens | |||
| 15. | ALA4865048 | 17 | EC50 | = | 160 | nM | ALA4841976 | 6.80 | nM | Homo sapiens | ||
| 16. | ALA4865048 | 17 | pEC50 | = | 6.8 | ALA4841976 | 6.80 | nM | Homo sapiens | |||
| 17. | ALA4865048 | 17 | Selectivity ratio | > | 7600 | ALA4841975 | ||||||
| 18. | ALA4865048 | 17 | Selectivity ratio | > | 7600 | ALA4841974 | ||||||
| 19. | ALA4865048 | 17 | Selectivity ratio | > | 7600 | ALA4841973 | ||||||
| 20. | ALA4865048 | 17 | Ki | > | 10 | nM | ALA4841972 | nM | Homo sapiens |
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