| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4865298 | 7 | permeability | = | 6.4 | 10^-6 cm/s | ALA4828038 | 10^-6 cm/s | ||||
| 2. | ALA4865298 | 7 | Ratio | = | 3.5 | ALA4828037 | ||||||
| 3. | ALA4865298 | 7 | PPB | = | 91.9 | % | ALA4828036 | % | ||||
| 4. | ALA4865298 | 7 | PPB | = | 94 | % | ALA4828035 | % | ||||
| 5. | ALA4865298 | 7 | t1/2 | = | 2.7 | hr | ALA4828034 | hr | ||||
| 6. | ALA4865298 | 7 | fVdss | = | 28 | L/Kg | ALA4828033 | L/Kg | ||||
| 7. | ALA4865298 | 7 | Vdss | = | 2.3 | L/Kg | ALA4828032 | L.kg-1 | ||||
| 8. | ALA4865298 | 7 | CL free | = | 123 | ml/min.Kg | ALA4828031 | mL.min-1.kg-1 | ||||
| 9. | ALA4865298 | 7 | CL | = | 10 | ml/min.Kg | ALA4828030 | mL.min-1.kg-1 | ||||
| 10. | ALA4865298 | 7 | Kinetic_solubility | = | 15 | uM | ALA4828024 | nM | ||||
| 11. | ALA4865298 | 7 | logD | = | 2.4 | ALA4828023 | ||||||
| 12. | ALA4865298 | 7 | fEC50 | = | 49 | nM | ALA4828022 | nM | Rattus norvegicus | |||
| 13. | ALA4865298 | 7 | IC50 | = | 14 | nM | ALA4828021 | 7.85 | nM | Rattus norvegicus | ||
| 14. | ALA4865298 | 7 | IC50 | = | 7.4 | nM | ALA4828020 | 8.13 | nM | Homo sapiens |
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