| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4865552 | 20aa | MIC | = | 3.63 | ug ml-1 | ALA4837711 | ug.mL-1 | Mycobacterium tuberculosis | |||
| 2. | ALA4865552 | 20aa | F | = | 128 | % | ALA4837710 | % | ||||
| 3. | ALA4865552 | 20aa | CL | = | 2.71 | ml/min.kg | ALA4837709 | mL.min-1.kg-1 | ||||
| 4. | ALA4865552 | 20aa | Vz | = | 0.762 | L/Kg | ALA4837708 | L.kg-1 | ||||
| 5. | ALA4865552 | 20aa | MRT | = | 5.86 | hr | ALA4837707 | hr | ||||
| 6. | ALA4865552 | 20aa | MRT | = | 4.71 | hr | ALA4837706 | hr | ||||
| 7. | ALA4865552 | 20aa | AUC | = | 78669 | hr.ng/ml | ALA4837705 | ng.hr.mL-1 | ||||
| 8. | ALA4865552 | 20aa | AUC | = | 6162 | hr.ng/ml | ALA4837704 | ng.hr.mL-1 | ||||
| 9. | ALA4865552 | 20aa | AUCt | = | 77649 | hr.ng/ml | ALA4837703 | ng.hr.mL-1 | ||||
| 10. | ALA4865552 | 20aa | AUCt | = | 6080 | hr.ng/ml | ALA4837702 | ng.hr.mL-1 | ||||
| 11. | ALA4865552 | 20aa | Cmax | = | 10253 | ng/ml | ALA4837701 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 12. | ALA4865552 | 20aa | Cmax | = | 1791 | ng/ml | ALA4837700 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 13. | ALA4865552 | 20aa | Tmax | = | 1.33 | hr | ALA4837699 | hr | ||||
| 14. | ALA4865552 | 20aa | beta t1/2 | = | 3.76 | hr | ALA4837698 | hr | ||||
| 15. | ALA4865552 | 20aa | beta t1/2 | = | 4.08 | hr | ALA4837697 | hr | ||||
| 16. | ALA4865552 | 20aa | IC50 | = | 6.07 | uM | ALA4837696 | 5.22 | nM | Homo sapiens | ||
| 17. | ALA4865552 | 20aa | IC50 | > | 50 | uM | ALA4837695 | nM | Homo sapiens | |||
| 18. | ALA4865552 | 20aa | IC50 | = | 1.63 | uM | ALA4837694 | 5.79 | nM | |||
| 19. | ALA4865552 | 20aa | IC50 | = | 17.82 | uM | ALA4837693 | 4.75 | nM | Homo sapiens | ||
| 20. | ALA4865552 | 20aa | IC50 | > | 64 | ug ml-1 | ALA4837692 | ug.mL-1 | Chlorocebus sabaeus |
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