| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4865816 | 40 | Activity | = | 266 | nM | ALA4809295 | nM | Homo sapiens | |||
| 2. | ALA4865816 | 40 | Activity | 0 | ALA4809292 | Not Active | Homo sapiens | |||||
| 3. | ALA4865816 | 40 | F | = | 100 | % | ALA4809291 | % | ||||
| 4. | ALA4865816 | 40 | t1/2 | = | 8.3 | hr | ALA4809290 | hr | ||||
| 5. | ALA4865816 | 40 | Vdss | = | 0.55 | L/Kg | ALA4809289 | L.kg-1 | ||||
| 6. | ALA4865816 | 40 | F | = | 78 | % | ALA4809288 | % | ||||
| 7. | ALA4865816 | 40 | t1/2 | = | 9.3 | hr | ALA4809287 | hr | ||||
| 8. | ALA4865816 | 40 | Vdss | = | 2.1 | L/Kg | ALA4809286 | L.kg-1 | ||||
| 9. | ALA4865816 | 40 | F | = | 100 | % | ALA4809285 | % | ||||
| 10. | ALA4865816 | 40 | t1/2 | = | 13 | hr | ALA4809284 | hr | ||||
| 11. | ALA4865816 | 40 | Vdss | = | 2 | L/Kg | ALA4809283 | L.kg-1 | ||||
| 12. | ALA4865816 | 40 | EC50 | = | 43 | nM | ALA4809280 | 7.37 | nM | |||
| 13. | ALA4865816 | 40 | CL | = | 0.05 | L/Kg.hr | ALA4809279 | L/Kg.hr | ||||
| 14. | ALA4865816 | 40 | CL | = | 0.38 | L/Kg.hr | ALA4809278 | L/Kg.hr | ||||
| 15. | ALA4865816 | 40 | CL | = | 0.17 | L/Kg.hr | ALA4809277 | L/Kg.hr | ||||
| 16. | ALA4865816 | 40 | Efficacy | = | 63 | % | ALA4809276 | % | Rattus norvegicus | |||
| 17. | ALA4865816 | 40 | MEC | = | 10 | nM | ALA4809275 | nM | Rattus norvegicus |
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