| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4866378 | 3d | INH | 0 | ALA4832695 | Not Active | % | |||||
| 2. | ALA4866378 | 3d | INH | 0 | ALA4832694 | Not Active | % | |||||
| 3. | ALA4866378 | 3d | INH | 0 | ALA4832693 | Not Active | % | |||||
| 4. | ALA4866378 | 3d | INH | 0 | ALA4832692 | Not Active | % | Homo sapiens | ||||
| 5. | ALA4866378 | 3d | CC50 | > | 100 | uM | ALA4832691 | nM | Homo sapiens | |||
| 6. | ALA4866378 | 3d | CC50 | 0 | ALA4832690 | Not Determined | Mus musculus | |||||
| 7. | ALA4866378 | 3d | EC50 | = | 1.4 | uM | ALA4832689 | 5.85 | nM | Trypanosoma brucei brucei | ||
| 8. | ALA4866378 | 3d | Activity | = | 47 | % | ALA4832686 | % | Trypanosoma brucei rhodesiense | |||
| 9. | ALA4866378 | 3d | Activity | 0 | ALA4832685 | Active | Trypanosoma brucei rhodesiense | |||||
| 10. | ALA4866378 | 3d | Ki | = | 25 | nM | ALA4832682 | 7.60 | nM | Trypanosoma brucei rhodesiense | ||
| 11. | ALA4866378 | 3d | Activity | 0 | ALA4832681 | Active | Trypanosoma brucei rhodesiense | |||||
| 12. | ALA4866378 | 3d | INH | = | 35 | % | ALA4832680 | % | Homo sapiens | |||
| 13. | ALA4866378 | 3d | Selectivity Index | = | 12 | ALA4832679 | ||||||
| 14. | ALA4866378 | 3d | Ki | = | 0.181 | uM | ALA4832676 | 6.74 | nM | Homo sapiens | ||
| 15. | ALA4866378 | 3d | Ki | = | 0.015 | uM | ALA4832674 | 7.82 | nM | Trypanosoma brucei rhodesiense |
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