# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | GLPG2938 | 40 | fIC50 | = | 0.6 | nM | ALA4836100 | nM | Homo sapiens | |||
2. | GLPG2938 | 40 | INH | 0 | ALA4836099 | Not Active | % | Homo sapiens | ||||
3. | GLPG2938 | 40 | Activity | 0 | ALA4836096 | Active | Mus musculus | |||||
4. | GLPG2938 | 40 | Activity | 0 | ALA4836095 | Active | Homo sapiens | |||||
5. | GLPG2938 | 40 | Therm_solubility | = | 23 | ug ml-1 | ALA4836091 | ug.mL-1 | ||||
6. | GLPG2938 | 40 | Therm_solubility | = | 2.7 | ug ml-1 | ALA4836090 | ug.mL-1 | ||||
7. | GLPG2938 | 40 | PPB | = | 99.7 | % | ALA4836089 | % | ||||
8. | GLPG2938 | 40 | PPB | > | 99.9 | % | ALA4836088 | % | ||||
9. | GLPG2938 | 40 | PPB | = | 99.9 | % | ALA4836087 | % | ||||
10. | GLPG2938 | 40 | F | = | 29 | % | ALA4836083 | % | ||||
11. | GLPG2938 | 40 | F | = | 64 | % | ALA4836082 | % | ||||
12. | GLPG2938 | 40 | Vdss | = | 1.1 | L/Kg | ALA4836081 | L.kg-1 | ||||
13. | GLPG2938 | 40 | Vdss | = | 0.35 | L/Kg | ALA4836080 | L.kg-1 | ||||
14. | GLPG2938 | 40 | Vdss | = | 0.81 | L/Kg | ALA4836079 | L.kg-1 | ||||
15. | GLPG2938 | 40 | CL | = | 0.1 | L/hr/kg | ALA4836078 | mL.min-1.kg-1 | ||||
16. | GLPG2938 | 40 | CL | = | 0.091 | L/hr/kg | ALA4836077 | mL.min-1.kg-1 | ||||
17. | GLPG2938 | 40 | CL | = | 0.24 | L/hr/kg | ALA4836076 | mL.min-1.kg-1 | ||||
18. | GLPG2938 | 40 | t1/2 | = | 7.6 | hr | ALA4836075 | hr | ||||
19. | GLPG2938 | 40 | t1/2 | = | 2.7 | hr | ALA4836074 | hr | ||||
20. | GLPG2938 | 40 | t1/2 | = | 2.3 | hr | ALA4836073 | hr |