| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4868638 | 7 | CL | = | 61.6 | ml/min.kg | ALA4806286 | mL.min-1.kg-1 | ||||
| 2. | ALA4868638 | 7 | %AUCextra | = | 1 | % | ALA4806285 | % | ||||
| 3. | ALA4868638 | 7 | AUC | = | 331817 | min.ng/ml | ALA4806284 | ng.hr.mL-1 | ||||
| 4. | ALA4868638 | 7 | AUClast | = | 10 | uM.hr | ALA4806283 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 5. | ALA4868638 | 7 | AUClast | = | 328306 | min.ng/ml | ALA4806283 | ng.hr.mL-1 | ||||
| 6. | ALA4868638 | 7 | Cmax | = | 2.7 | uM | ALA4806282 | nM | ||||
| 7. | ALA4868638 | 7 | Cmax | = | 1430 | ng/ml | ALA4806282 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 8. | ALA4868638 | 7 | Tmax | = | 1 | hr | ALA4806281 | hr | ||||
| 9. | ALA4868638 | 7 | t1/2 | = | 3.71 | hr | ALA4806280 | hr | ||||
| 10. | ALA4868638 | 7 | INH | = | 54 | % | ALA4806279 | % | Homo sapiens | |||
| 11. | ALA4868638 | 7 | INH | = | 29 | % | ALA4806278 | % | Homo sapiens | |||
| 12. | ALA4868638 | 7 | INH | = | 54 | % | ALA4806277 | % | Homo sapiens | |||
| 13. | ALA4868638 | 7 | INH | = | 39 | % | ALA4806276 | % | Homo sapiens | |||
| 14. | ALA4868638 | 7 | t1/2 | = | 25 | min | ALA4806275 | hr | ||||
| 15. | ALA4868638 | 7 | t1/2 | = | 18 | min | ALA4806274 | hr | ||||
| 16. | ALA4868638 | 7 | t1/2 | = | 27 | min | ALA4806273 | hr | ||||
| 17. | ALA4868638 | 7 | solubility | = | 0.7 | uM | ALA4806272 | nM | ||||
| 18. | ALA4868638 | 7 | GI50 | = | 51 | nM | ALA4806271 | nM | Homo sapiens | |||
| 19. | ALA4868638 | 7 | GI50 | = | 78 | nM | ALA4806270 | nM | Homo sapiens | |||
| 20. | ALA4868638 | 7 | IC50 | = | 253 | nM | ALA4806269 | 6.60 | nM |
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