# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4868958 | 4 | INH | = | 89 | % | ALA4806279 | % | Homo sapiens | |||
2. | ALA4868958 | 4 | INH | = | 57 | % | ALA4806278 | % | Homo sapiens | |||
3. | ALA4868958 | 4 | INH | = | 99 | % | ALA4806277 | % | Homo sapiens | |||
4. | ALA4868958 | 4 | INH | = | 97 | % | ALA4806276 | % | Homo sapiens | |||
5. | ALA4868958 | 4 | t1/2 | = | 9 | min | ALA4806275 | hr | ||||
6. | ALA4868958 | 4 | t1/2 | = | 6 | min | ALA4806274 | hr | ||||
7. | ALA4868958 | 4 | t1/2 | = | 16 | min | ALA4806273 | hr | ||||
8. | ALA4868958 | 4 | solubility | = | 0.8 | uM | ALA4806272 | nM | ||||
9. | ALA4868958 | 4 | GI50 | < | 2 | nM | ALA4806271 | nM | Homo sapiens | |||
10. | ALA4868958 | 4 | GI50 | < | 2 | nM | ALA4806270 | nM | Homo sapiens | |||
11. | ALA4868958 | 4 | IC50 | = | 215 | nM | ALA4806269 | 6.67 | nM | |||
12. | ALA4868958 | 4 | Kd | = | 6 | nM | ALA4806268 | 8.22 | nM | Homo sapiens | ||
13. | ALA4868958 | 4 | Kd | = | 18 | nM | ALA4806267 | 7.75 | nM | Homo sapiens | ||
14. | ALA4868958 | 4 | IC50 | = | 1279 | nM | ALA4806266 | 5.89 | nM | Homo sapiens | ||
15. | ALA4868958 | 4 | IC50 | = | 870 | nM | ALA4806265 | 6.06 | nM | Homo sapiens |