| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4869361 | AQU-019 | Activity | = | 15 | % | ALA4829082 | % | Rattus norvegicus | |||
| 2. | ALA4869361 | AQU-019 | Activity | = | 15 | % | ALA4829081 | % | Rattus norvegicus | |||
| 3. | ALA4869361 | AQU-019 | Activity | 0 | ALA4829072 | Not Active | Rattus norvegicus | |||||
| 4. | ALA4869361 | AQU-019 | Activity | = | 8 | % | ALA4829071 | % | Rattus norvegicus | |||
| 5. | ALA4869361 | AQU-019 | Activity | = | 15 | % | ALA4829070 | % | Rattus norvegicus | |||
| 6. | ALA4869361 | AQU-019 | Tmax | = | 0.75 | hr | ALA4829069 | hr | ||||
| 7. | ALA4869361 | AQU-019 | Cmax | = | 362 | ng/ml | ALA4829068 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 8. | ALA4869361 | AQU-019 | betat1/2(app) | = | 1.22 | hr | ALA4829067 | hr | ||||
| 9. | ALA4869361 | AQU-019 | AUC | = | 705 | ng.hr/ml | ALA4829066 | ng.hr.mL-1 | ||||
| 10. | ALA4869361 | AQU-019 | AUCt | = | 697 | ng.hr/ml | ALA4829065 | ng.hr.mL-1 | ||||
| 11. | ALA4869361 | AQU-019 | Stability | = | 99 | % | ALA4829064 | % | ||||
| 12. | ALA4869361 | AQU-019 | IC50 | > | 100000 | nM | ALA4829063 | nM | Homo sapiens | |||
| 13. | ALA4869361 | AQU-019 | IC50 | = | 4.8 | nM | ALA4829062 | 8.32 | nM | Homo sapiens | ||
| 14. | ALA4869361 | AQU-019 | IC50 | > | 100000 | nM | ALA4829061 | nM | Homo sapiens | |||
| 15. | ALA4869361 | AQU-019 | IC50 | > | 100000 | nM | ALA4829060 | nM | Homo sapiens | |||
| 16. | ALA4869361 | AQU-019 | IC50 | > | 100000 | nM | ALA4829059 | nM | Homo sapiens | |||
| 17. | ALA4869361 | AQU-019 | IC50 | > | 100000 | nM | ALA4829058 | nM | Homo sapiens | |||
| 18. | ALA4869361 | AQU-019 | IC50 | = | 98000 | nM | ALA4829057 | 4.01 | nM | Homo sapiens | ||
| 19. | ALA4869361 | AQU-019 | IC50 | = | 74000 | nM | ALA4829056 | 4.13 | nM | Homo sapiens | ||
| 20. | ALA4869361 | AQU-019 | IC50 | = | 1000 | nM | ALA4829055 | 6.00 | nM | Homo sapiens |
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