# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4869882 | 20 | t1/2 | > | 1000 | min | ALA4822237 | hr | ||||
2. | ALA4869882 | 20 | t1/2 | = | 48 | min | ALA4822236 | hr | ||||
3. | ALA4869882 | 20 | t1/2 | = | 131 | min | ALA4822235 | hr | ||||
4. | ALA4869882 | 20 | t1/2 | = | 475 | min | ALA4822234 | hr | ||||
5. | ALA4869882 | 20 | PPB | = | 97.1 | % | ALA4822233 | % | ||||
6. | ALA4869882 | 20 | PPB | = | 97.2 | % | ALA4822232 | % | ||||
7. | ALA4869882 | 20 | PPB | = | 97.2 | % | ALA4822231 | % | ||||
8. | ALA4869882 | 20 | PPB | = | 97.6 | % | ALA4822230 | % | ||||
9. | ALA4869882 | 20 | Ratio | = | 4.6 | ALA4822229 | ||||||
10. | ALA4869882 | 20 | permeability | = | 14 | 10^-6 cm/s | ALA4822228 | 10^-6 cm/s | ||||
11. | ALA4869882 | 20 | solubility | = | 37 | uM | ALA4822227 | nM | ||||
12. | ALA4869882 | 20 | IC50 | = | 0.027 | uM | ALA4822226 | 7.57 | nM | Homo sapiens | ||
13. | ALA4869882 | 20 | IC50 | = | 0.003 | uM | ALA4822225 | 8.52 | nM | Homo sapiens |