# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4870168 | 23 | Stability | 0 | ALA4841991 | Stable | % | |||||
2. | ALA4870168 | 23 | t1/2 | = | 7.9 | hr | ALA4841990 | hr | ||||
3. | ALA4870168 | 23 | Stability | = | 3 | % | ALA4841989 | % | ||||
4. | ALA4870168 | 23 | Stability | = | 67 | % | ALA4841988 | % | ||||
5. | ALA4870168 | 23 | Stability | = | 87 | % | ALA4841987 | % | ||||
6. | ALA4870168 | 23 | Stability | 0 | ALA4841986 | Not Determined | % | |||||
7. | ALA4870168 | 23 | Stability | = | 94 | % | ALA4841985 | % | ||||
8. | ALA4870168 | 23 | Intrinsic activity | = | 0.95 | % | ALA4841983 | % | Homo sapiens | |||
9. | ALA4870168 | 23 | pEC50 | = | 7.92 | ALA4841982 | 7.92 | nM | Homo sapiens | |||
10. | ALA4870168 | 23 | Intrinsic activity | = | 0.67 | % | ALA4841981 | % | Homo sapiens | |||
11. | ALA4870168 | 23 | pEC50 | = | 6.98 | ALA4841980 | 6.98 | nM | Homo sapiens | |||
12. | ALA4870168 | 23 | Intrinsic activity | = | 0.76 | % | ALA4841979 | % | Homo sapiens | |||
13. | ALA4870168 | 23 | pEC50 | = | 6.79 | ALA4841978 | 6.79 | nM | Homo sapiens | |||
14. | ALA4870168 | 23 | Intrinsic activity | = | 0.67 | % | ALA4841977 | % | Homo sapiens | |||
15. | ALA4870168 | 23 | EC50 | = | 120 | nM | ALA4841976 | 6.92 | nM | Homo sapiens | ||
16. | ALA4870168 | 23 | pEC50 | = | 6.94 | ALA4841976 | 6.94 | nM | Homo sapiens | |||
17. | ALA4870168 | 23 | Selectivity ratio | > | 4700 | ALA4841975 | ||||||
18. | ALA4870168 | 23 | Selectivity ratio | > | 1400 | ALA4841974 | ||||||
19. | ALA4870168 | 23 | Selectivity ratio | > | 4700 | ALA4841973 | ||||||
20. | ALA4870168 | 23 | Ki | > | 10 | nM | ALA4841972 | nM | Homo sapiens |