# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4870760 | 16c | Selectivity Index | > | 3.3 | ALA4822816 | ||||||
2. | ALA4870760 | 16c | IC50 | > | 100 | uM | ALA4822815 | nM | Chlorocebus sabaeus | |||
3. | ALA4870760 | 16c | IC50 | > | 100 | uM | ALA4822814 | nM | Homo sapiens | |||
4. | ALA4870760 | 16c | IC50 | = | 30.2 | uM | ALA4822813 | 4.52 | nM | Homo sapiens | ||
5. | ALA4870760 | 16c | Efficacy | = | 8 | % | ALA4822812 | % | Homo sapiens | |||
6. | ALA4870760 | 16c | Efficacy | = | 29 | % | ALA4822811 | % | Homo sapiens | |||
7. | ALA4870760 | 16c | Efficacy | = | 68 | % | ALA4822808 | % | Homo sapiens | |||
8. | ALA4870760 | 16c | EC50 | = | 1.009 | uM | ALA4822806 | 6.00 | nM | Homo sapiens | ||
9. | ALA4870760 | 16c | Selectivity ratio | = | 31.05 | ALA4822804 | ||||||
10. | ALA4870760 | 16c | Ki | = | 2615.38 | nM | ALA4822803 | 5.58 | nM | Homo sapiens | ||
11. | ALA4870760 | 16c | Ki | = | 84.24 | nM | ALA4822802 | 7.07 | nM | Homo sapiens | ||
12. | ALA4870760 | 16c | Selectivity ratio | = | 28.31 | ALA4822801 | ||||||
13. | ALA4870760 | 16c | RBA | = | 0.13 | % | ALA4822800 | % | Homo sapiens | |||
14. | ALA4870760 | 16c | RBA | = | 3.68 | % | ALA4822799 | % | Homo sapiens |