# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4870914 | 5f | MRT | = | 2.42 | hr | ALA4831402 | hr | ||||
2. | ALA4870914 | 5f | AUC | = | 2707 | hr.ng/ml | ALA4831401 | ng.hr.mL-1 | ||||
3. | ALA4870914 | 5f | AUCt | = | 2523 | hr.ng/ml | ALA4831400 | ng.hr.mL-1 | ||||
4. | ALA4870914 | 5f | Cmax | = | 1691 | ng/ml | ALA4831399 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
5. | ALA4870914 | 5f | Tmax | = | 0.25 | hr | ALA4831398 | hr | ||||
6. | ALA4870914 | 5f | t1/2 | = | 2.38 | hr | ALA4831397 | hr | ||||
7. | ALA4870914 | 5f | INH | = | 58.5 | % | ALA4831396 | % | Homo sapiens | |||
8. | ALA4870914 | 5f | IC50 | = | 0.63 | uM | ALA4831395 | 6.20 | nM | Homo sapiens | ||
9. | ALA4870914 | 5f | IC50 | = | 0.25 | uM | ALA4831394 | 6.60 | nM | Homo sapiens | ||
10. | ALA4870914 | 5f | IC50 | = | 24.3 | nM | ALA4831392 | 7.61 | nM | Homo sapiens |