| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4871803 | 10 | INH | = | 75 | % | ALA4844323 | % | Homo sapiens | |||
| 2. | ALA4871803 | 10 | INH | = | 75 | % | ALA4844322 | % | Homo sapiens | |||
| 3. | ALA4871803 | 10 | INH | > | 90 | % | ALA4844321 | % | Homo sapiens | |||
| 4. | ALA4871803 | 10 | INH | > | 90 | % | ALA4844320 | % | Homo sapiens | |||
| 5. | ALA4871803 | 10 | INH | > | 90 | % | ALA4844319 | % | Homo sapiens | |||
| 6. | ALA4871803 | 10 | INH | > | 90 | % | ALA4844318 | % | Homo sapiens | |||
| 7. | ALA4871803 | 10 | PPB | = | 73 | % | ALA4844317 | % | ||||
| 8. | ALA4871803 | 10 | AUC | = | 35 | uM.hr | ALA4844316 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 9. | ALA4871803 | 10 | AUC | = | 27 | uM.hr | ALA4844315 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 10. | ALA4871803 | 10 | CL | < | 38 | ml/min.kg | ALA4844313 | mL.min-1.kg-1 | ||||
| 11. | ALA4871803 | 10 | CL | = | 20 | ml/min.kg | ALA4844308 | mL.min-1.kg-1 | ||||
| 12. | ALA4871803 | 10 | PPB | = | 53 | % | ALA4844307 | % | ||||
| 13. | ALA4871803 | 10 | logD | = | 2 | ALA4844306 | ||||||
| 14. | ALA4871803 | 10 | IC50 | = | 317 | nM | ALA4844305 | 6.50 | nM | Homo sapiens | ||
| 15. | ALA4871803 | 10 | IC50 | = | 4.8 | nM | ALA4844304 | 8.32 | nM | Homo sapiens |
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