| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4872783 | 29; K1600 | Drug uptake | = | 326 | nM | ALA4818734 | nM | ||||
| 2. | ALA4872783 | 29; K1600 | Cp | = | 207 | nM | ALA4818733 | nM | ||||
| 3. | ALA4872783 | 29; K1600 | Drug uptake | = | 2315 | nM | ALA4818732 | nM | ||||
| 4. | ALA4872783 | 29; K1600 | IC50 | = | 51.02 | uM | ALA4818731 | 4.29 | nM | Rattus norvegicus | ||
| 5. | ALA4872783 | 29; K1600 | IC50 | = | 49.31 | uM | ALA4818730 | 4.31 | nM | Homo sapiens | ||
| 6. | ALA4872783 | 29; K1600 | Selectivity Index | = | 1.76 | ALA4818729 | ||||||
| 7. | ALA4872783 | 29; K1600 | INH | = | 68.84 | % | ALA4818728 | % | Rattus norvegicus | |||
| 8. | ALA4872783 | 29; K1600 | INH | = | 77.59 | % | ALA4818727 | % | Homo sapiens | |||
| 9. | ALA4872783 | 29; K1600 | IC50 | = | 7.24 | uM | ALA4818726 | 5.14 | nM | Rattus norvegicus | ||
| 10. | ALA4872783 | 29; K1600 | IC50 | = | 4.7 | uM | ALA4818724 | 5.33 | nM | Homo sapiens | ||
| 11. | ALA4872783 | 29; K1600 | Cp | = | 1673 | nM | ALA4818723 | nM | ||||
| 12. | ALA4872783 | 29; K1600 | BBR | = | 138 | ALA4818721 | ||||||
| 13. | ALA4872783 | 29; K1600 | IC50 | = | 17.6 | uM | ALA4818720 | 4.75 | nM | Homo sapiens | ||
| 14. | ALA4872783 | 29; K1600 | IC50 | = | 10 | uM | ALA4818719 | 5.00 | nM | Homo sapiens |
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