# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4873416 | 9 | Imax | > | 99 | % | ALA4843621 | % | Homo sapiens | |||
2. | ALA4873416 | 9 | IC50 | = | 9 | nM | ALA4843620 | 8.05 | nM | Homo sapiens | ||
3. | ALA4873416 | 9 | Activity | = | 31 | mg/dl | ALA4843614 | mg/dl | ||||
4. | ALA4873416 | 9 | F | = | 65 | % | ALA4843613 | % | ||||
5. | ALA4873416 | 9 | t1/2 | = | 2.5 | hr | ALA4843612 | hr | ||||
6. | ALA4873416 | 9 | CL | = | 18 | ml/min.kg | ALA4843610 | mL.min-1.kg-1 | ||||
7. | ALA4873416 | 9 | AUC/dose | = | 0.86 | uM.hr.Kg/mg | ALA4843608 | uM.hr.Kg/mg | ||||
8. | ALA4873416 | 9 | Cmax | = | 0.43 | uM | ALA4843607 | nM | ||||
9. | ALA4873416 | 9 | solubility | = | 16 | uM | ALA4843605 | nM | ||||
10. | ALA4873416 | 9 | IC50 | = | 10 | uM | ALA4843604 | 5.00 | nM | Homo sapiens | ||
11. | ALA4873416 | 9 | Emax | = | 0 | % | ALA4843603 | % | Homo sapiens | |||
12. | ALA4873416 | 9 | EC50 | > | 30 | uM | ALA4843602 | nM | Homo sapiens |