# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4874732 | (R)-2i | IC50 | = | 67.3 | uM | ALA4829570 | 4.17 | nM | Homo sapiens | ||
2. | ALA4874732 | (R)-2i | INH | = | 79.7 | % | ALA4829569 | % | Homo sapiens | |||
3. | ALA4874732 | (R)-2i | INH | = | 38.6 | % | ALA4829568 | % | Homo sapiens | |||
4. | ALA4874732 | (R)-2i | INH | = | 7.7 | % | ALA4829567 | % | Homo sapiens | |||
5. | ALA4874732 | (R)-2i | Activity | 0 | ALA4829566 | Not Active | Homo sapiens | |||||
6. | ALA4874732 | (R)-2i | Activity | = | 3794 | umol/L | ALA4829565 | umol/L | Rattus norvegicus | |||
7. | ALA4874732 | (R)-2i | Activity | = | 124 | U/mg | ALA4829564 | U/mg | Rattus norvegicus | |||
8. | ALA4874732 | (R)-2i | Activity | = | 47 | nmol/ml | ALA4829563 | nmol/ml | Rattus norvegicus | |||
9. | ALA4874732 | (R)-2i | Activity | = | 132 | U/L | ALA4829562 | U/L | Rattus norvegicus | |||
10. | ALA4874732 | (R)-2i | Survival | = | 51.9 | % | ALA4829559 | % | Rattus norvegicus | |||
11. | ALA4874732 | (R)-2i | Survival | = | 53 | % | ALA4829558 | % | Rattus norvegicus | |||
12. | ALA4874732 | (R)-2i | Survival | = | 58.2 | % | ALA4829557 | % | Rattus norvegicus | |||
13. | ALA4874732 | (R)-2i | Survival | = | 58 | % | ALA4829556 | % | Rattus norvegicus | |||
14. | ALA4874732 | (R)-2i | Survival | = | 66.6 | % | ALA4829555 | % | Rattus norvegicus | |||
15. | ALA4874732 | (R)-2i | Survival | = | 60.1 | % | ALA4829554 | % | Rattus norvegicus | |||
16. | ALA4874732 | (R)-2i | Survival | <= | 96 | % | ALA4829553 | % | Rattus norvegicus | |||
17. | ALA4874732 | (R)-2i | Survival | = | 67 | % | ALA4829550 | % | Rattus norvegicus | |||
18. | ALA4874732 | (R)-2i | Survival | = | 60 | % | ALA4829549 | % | Rattus norvegicus |