# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | Activity | 0 | ALA4821556 | Active | ||||||
2. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | Activity | 0 | ALA4821555 | Active | ||||||
3. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | Activity | 0 | ALA4821554 | Active | ||||||
4. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | Activity | 0 | ALA4821553 | Active | ||||||
5. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | Activity | 0 | ALA4821552 | Active | ||||||
6. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | Activity | 0 | ALA4821551 | Non-Toxic | ||||||
7. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | Activity | 0 | ALA4821550 | Active | Homo sapiens | |||||
8. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | INH | > | 50 | % | ALA4821548 | % | Homo sapiens | |||
9. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | INH | > | 50 | % | ALA4821547 | % | Homo sapiens | |||
10. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | Activity | 0 | ALA4821546 | Non-Toxic | ||||||
11. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | Activity | 0 | ALA4821545 | Toxic | ||||||
12. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | Activity | 0 | ALA4821544 | Active | Homo sapiens | |||||
13. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | Activity | 0 | ALA4821543 | Active | Homo sapiens | |||||
14. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | INH | = | 55 | % | ALA4821542 | % | Homo sapiens | |||
15. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | Activity | 0 | ALA4821541 | Dose-Dependent Effect | Homo sapiens | |||||
16. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | LC50 | = | 4.71 | uM | ALA4821540 | nM | Homo sapiens | |||
17. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | TGI | = | 1.65 | uM | ALA4821540 | nM | Homo sapiens | |||
18. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | GI50 | = | 0.4 | uM | ALA4821540 | nM | Homo sapiens | |||
19. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | LC50 | = | 5.46 | uM | ALA4821539 | nM | Homo sapiens | |||
20. | ALA4874753 | 22d; GL0388, , Diastereomeric mixture 50:50 | TGI | = | 2.54 | uM | ALA4821539 | nM | Homo sapiens |