# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4875730 | 6'k | Cmax | = | 46.6 | ng/ml | ALA4831826 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
2. | ALA4875730 | 6'k | Tmax | = | 0.57 | hr | ALA4831825 | hr | ||||
3. | ALA4875730 | 6'k | t1/2 | = | 3.93 | hr | ALA4831824 | hr | ||||
4. | ALA4875730 | 6'k | MRT(t) | = | 2.68 | hr | ALA4831823 | hr | ||||
5. | ALA4875730 | 6'k | AUC | = | 153 | hr.ng/ml | ALA4831822 | ng.hr.mL-1 | ||||
6. | ALA4875730 | 6'k | Activity | = | 44 | % | ALA4831821 | % | Homo sapiens | |||
7. | ALA4875730 | 6'k | Activity | 0 | ALA4831820 | Non-Toxic | ||||||
8. | ALA4875730 | 6'k | Activity | 0 | ALA4831819 | Non-Toxic | ||||||
9. | ALA4875730 | 6'k | GI50 | = | 8.17 | uM | ALA4831814 | nM | Homo sapiens | |||
10. | ALA4875730 | 6'k | GI50 | = | 5.46 | uM | ALA4831813 | nM | ||||
11. | ALA4875730 | 6'k | GI50 | = | 6.73 | uM | ALA4831812 | nM | Homo sapiens | |||
12. | ALA4875730 | 6'k | GI50 | = | 4.71 | uM | ALA4831811 | nM | Homo sapiens | |||
13. | ALA4875730 | 6'k | GI50 | = | 0.76 | uM | ALA4831810 | nM | Homo sapiens | |||
14. | ALA4875730 | 6'k | IC50 | = | 40.6 | nM | ALA4831809 | 7.39 | nM | Homo sapiens | ||
15. | ALA4875730 | 6'k | GI50 | = | 0.35 | uM | ALA4831808 | nM | Homo sapiens | |||
16. | ALA4875730 | 6'k | INH | = | 102 | % | ALA4831807 | % | Homo sapiens |