# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4876602 | (R)-28 | Activity | = | 5.97 | % | ALA4811583 | % | Homo sapiens | |||
2. | ALA4876602 | (R)-28 | Activity | = | 9.92 | % | ALA4811582 | % | Homo sapiens | |||
3. | ALA4876602 | (R)-28 | Activity | = | 85.7 | % | ALA4811581 | % | Homo sapiens | |||
4. | ALA4876602 | (R)-28 | INH | 0 | ALA4811580 | Active | % | Homo sapiens | ||||
5. | ALA4876602 | (R)-28 | Cmax | = | 0.3 | uM | ALA4811577 | nM | ||||
6. | ALA4876602 | (R)-28 | t1/2 | = | 0.5 | hr | ALA4811576 | hr | ||||
7. | ALA4876602 | (R)-28 | AUC | = | 0.7 | uM.hr | ALA4811575 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
8. | ALA4876602 | (R)-28 | INH | = | 71 | % | ALA4811568 | % | Homo sapiens | |||
9. | ALA4876602 | (R)-28 | INH | 0 | ALA4811568 | Active | % | Homo sapiens | ||||
10. | ALA4876602 | (R)-28 | t1/2 | = | 8 | min | ALA4811567 | hr | ||||
11. | ALA4876602 | (R)-28 | IC50 | = | 0.034 | uM | ALA4811566 | 7.47 | nM | Homo sapiens | ||
12. | ALA4876602 | (R)-28 | IC50 | = | 0.04 | uM | ALA4811565 | 7.40 | nM | Homo sapiens | ||
13. | ALA4876602 | (R)-28 | IC50 | = | 0.07 | uM | ALA4811564 | 7.16 | nM | Homo sapiens |