# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4876736 | 26 | Stabilty | 0 | ALA4808914 | Stable | % | |||||
2. | ALA4876736 | 26 | solubility | > | 500 | uM | ALA4808913 | nM | ||||
3. | ALA4876736 | 26 | AUC | = | 209 | hr.nM | ALA4808911 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
4. | ALA4876736 | 26 | Cmax | = | 261 | nM | ALA4808909 | nM | ||||
5. | ALA4876736 | 26 | t1/2 | = | 30.7 | min | ALA4808907 | hr | ||||
6. | ALA4876736 | 26 | Activity | 0 | ALA4808906 | Non-Toxic | ||||||
7. | ALA4876736 | 26 | INH | 0 | ALA4808903 | Active | % | |||||
8. | ALA4876736 | 26 | INH | = | 1 | % | ALA4808902 | % | Mus musculus | |||
9. | ALA4876736 | 26 | IC50 | > | 1000 | nM | ALA4808901 | nM | Mus musculus | |||
10. | ALA4876736 | 26 | INH | = | 10 | % | ALA4808900 | % | Mus musculus | |||
11. | ALA4876736 | 26 | IC50 | > | 1000 | nM | ALA4808899 | nM | Mus musculus | |||
12. | ALA4876736 | 26 | IC50 | = | 23.1 | nM | ALA4808898 | 7.64 | nM | Mus musculus | ||
13. | ALA4876736 | 26 | INH | = | 92 | % | ALA4808897 | % | Mus musculus | |||
14. | ALA4876736 | 26 | INH | = | 8 | % | ALA4808896 | % | Homo sapiens | |||
15. | ALA4876736 | 26 | IC50 | > | 1000 | nM | ALA4808895 | nM | Homo sapiens | |||
16. | ALA4876736 | 26 | INH | = | 20 | % | ALA4808894 | % | Homo sapiens | |||
17. | ALA4876736 | 26 | IC50 | > | 1000 | nM | ALA4808893 | nM | Homo sapiens | |||
18. | ALA4876736 | 26 | INH | = | 99 | % | ALA4808892 | % | Homo sapiens | |||
19. | ALA4876736 | 26 | IC50 | = | 12.1 | nM | ALA4808886 | 7.92 | nM | Homo sapiens | ||
20. | ALA4876736 | 26 | IC50 | = | 9 | nM | ALA4808885 | 8.05 | nM | Homo sapiens |