| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4877264 | 10 | INH | 0 | ALA4834338 | Active | % | Mus musculus | ||||
| 2. | ALA4877264 | 10 | Activity | 0 | ALA4834337 | Active | Mus musculus | |||||
| 3. | ALA4877264 | 10 | Activity | 0 | ALA4834336 | Non-Toxic | ||||||
| 4. | ALA4877264 | 10 | Activity | 0 | ALA4834335 | Non-Toxic | ||||||
| 5. | ALA4877264 | 10 | fCmax | = | 6.8 | uM | ALA4834329 | uM | ||||
| 6. | ALA4877264 | 10 | fAUC | = | 41 | uM.hr | ALA4834326 | uM.hr | ||||
| 7. | ALA4877264 | 10 | Cmax | = | 19 | uM | ALA4834323 | nM | ||||
| 8. | ALA4877264 | 10 | AUC | = | 115 | uM.hr | ALA4834320 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 9. | ALA4877264 | 10 | PPB | = | 64.4 | % | ALA4834319 | % | ||||
| 10. | ALA4877264 | 10 | IC50 | = | 7.9 | uM | ALA4834318 | 5.10 | nM | Homo sapiens | ||
| 11. | ALA4877264 | 10 | IC50 | = | 19 | uM | ALA4834317 | 4.72 | nM | Homo sapiens | ||
| 12. | ALA4877264 | 10 | IC50 | = | 0.046 | uM | ALA4834316 | 7.34 | nM | Homo sapiens | ||
| 13. | ALA4877264 | 10 | Ratio | = | 0.03 | ALA4834315 | ||||||
| 14. | ALA4877264 | 10 | Ratio | = | 0.03 | ALA4834314 | ||||||
| 15. | ALA4877264 | 10 | F | = | 48 | % | ALA4834313 | % | ||||
| 16. | ALA4877264 | 10 | Cmax | = | 3.8 | uM | ALA4834311 | nM | ||||
| 17. | ALA4877264 | 10 | Cmax | = | 5.1 | uM | ALA4834310 | nM | ||||
| 18. | ALA4877264 | 10 | AUC | = | 12 | uM.hr | ALA4834307 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 19. | ALA4877264 | 10 | AUC | = | 5 | uM.hr | ALA4834306 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 20. | ALA4877264 | 10 | t1/2 | = | 2.4 | hr | ALA4834303 | hr |
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