# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4877388 | 6c | Activity | 0 | ALA4827170 | Not Active | ||||||
2. | ALA4877388 | 6c | Time | > | 60 | day | ALA4827168 | hr | Trypanosoma brucei rhodesiense | |||
3. | ALA4877388 | 6c | Selectivity Index | = | 1616 | ALA4827167 | ||||||
4. | ALA4877388 | 6c | Selectivity Index | = | 441.4 | ALA4827166 | ||||||
5. | ALA4877388 | 6c | IC50 | = | 11.2 | nM | ALA4827165 | 7.95 | nM | Plasmodium falciparum | ||
6. | ALA4877388 | 6c | IC50 | = | 41 | nM | ALA4827164 | 7.39 | nM | Trypanosoma brucei rhodesiense | ||
7. | ALA4877388 | 6c | deltaTm | = | 1 | degrees C | ALA4827163 | degrees C | ||||
8. | ALA4877388 | 6c | IC50 | = | 18.1 | uM | ALA4827162 | 4.74 | nM | Rattus norvegicus |