| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4877968 | 19 | F | = | 48 | % | ALA4810904 | % | ||||
| 2. | ALA4877968 | 19 | t1/2 | = | 11 | hr | ALA4810902 | hr | ||||
| 3. | ALA4877968 | 19 | Vdss | = | 9.6 | L/Kg | ALA4810901 | L.kg-1 | ||||
| 4. | ALA4877968 | 19 | CL | = | 10.2 | ml/min.kg | ALA4810900 | mL.min-1.kg-1 | ||||
| 5. | ALA4877968 | 19 | CLH | = | 44 | ml/min.kg | ALA4810899 | mL.min-1.kg-1 | ||||
| 6. | ALA4877968 | 19 | CLH | = | 55 | ml/min.kg | ALA4810898 | mL.min-1.kg-1 | ||||
| 7. | ALA4877968 | 19 | IC50 | = | 17 | nM | ALA4810897 | 7.77 | nM | Homo sapiens | ||
| 8. | ALA4877968 | 19 | Kinetic_solubility | = | 135 | uM | ALA4810894 | nM | ||||
| 9. | ALA4877968 | 19 | Papp | = | 5 | 10^-6 cm/s | ALA4810891 | 10^-6 cm/s | ||||
| 10. | ALA4877968 | 19 | Papp | = | 4 | 10^-6 cm/s | ALA4810890 | 10^-6 cm/s | ||||
| 11. | ALA4877968 | 19 | logD | = | 2.5 | ALA4810889 | ||||||
| 12. | ALA4877968 | 19 | IC50 | = | 0.4 | nM | ALA4810888 | 9.40 | nM | Homo sapiens | ||
| 13. | ALA4877968 | 19 | %max | = | 93 | % | ALA4810887 | % | Homo sapiens | |||
| 14. | ALA4877968 | 19 | DC50 | = | 0.19 | nM | ALA4810886 | nM | Homo sapiens |
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