# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4878039 | 28k; S62798 | Ratio | = | 1 | ALA4835338 | ||||||
2. | ALA4878039 | 28k; S62798 | Fabs | = | 66 | % | ALA4835337 | % | ||||
3. | ALA4878039 | 28k; S62798 | INH | = | 61 | % | ALA4835336 | % | Rattus norvegicus | |||
4. | ALA4878039 | 28k; S62798 | EC50 | = | 389 | nM | ALA4835334 | 6.41 | nM | Rattus norvegicus | ||
5. | ALA4878039 | 28k; S62798 | INH | = | 57 | % | ALA4835333 | % | Rattus norvegicus | |||
6. | ALA4878039 | 28k; S62798 | Ratio Ki | = | 300000 | ALA4835332 | ||||||
7. | ALA4878039 | 28k; S62798 | Ratio Ki | = | 7000 | ALA4835331 | ||||||
8. | ALA4878039 | 28k; S62798 | CL | = | 9.84 | ml/min.kg | ALA4835330 | mL.min-1.kg-1 | ||||
9. | ALA4878039 | 28k; S62798 | beta t1/2 | = | 0.47 | hr | ALA4835329 | hr | ||||
10. | ALA4878039 | 28k; S62798 | AUC | = | 3.88 | micromol.hr/L | ALA4835328 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
11. | ALA4878039 | 28k; S62798 | Ki | = | 282 | uM | ALA4835327 | nM | Homo sapiens | |||
12. | ALA4878039 | 28k; S62798 | Stabilty | = | 85 | % | ALA4835326 | % | ||||
13. | ALA4878039 | 28k; S62798 | Stabilty | = | 100 | % | ALA4835325 | % | ||||
14. | ALA4878039 | 28k; S62798 | Stabilty | = | 100 | % | ALA4835324 | % | ||||
15. | ALA4878039 | 28k; S62798 | Stabilty | = | 100 | % | ALA4835323 | % | ||||
16. | ALA4878039 | 28k; S62798 | Stabilty | = | 100 | % | ALA4835322 | % | ||||
17. | ALA4878039 | 28k; S62798 | Stabilty | = | 100 | % | ALA4835321 | % | ||||
18. | ALA4878039 | 28k; S62798 | CL | = | 9.54 | ml/min.kg | ALA4835320 | mL.min-1.kg-1 | ||||
19. | ALA4878039 | 28k; S62798 | Vdss | = | 0.3 | L/Kg | ALA4835319 | L.kg-1 | ||||
20. | ALA4878039 | 28k; S62798 | Fu | = | 95 | % | ALA4835318 |