| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4878072 | Senexin C/6148/GJ-2331/2335 | Ratio | = | 5 | ALA4805272 | ||||||
| 2. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | Activity | 0 | ALA4805270 | Active | Mus musculus | |||||
| 3. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | Drug uptake | 0 | ALA4805269 | Active | ||||||
| 4. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | Activity | 0 | ALA4805268 | Active | Homo sapiens | |||||
| 5. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | t1/2 | = | 3.8 | hr | ALA4805267 | hr | ||||
| 6. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | AUC | = | 817 | ng.hr/ml | ALA4805266 | ng.hr.mL-1 | ||||
| 7. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | IC50 | = | 82 | nM | ALA4805265 | 7.09 | nM | |||
| 8. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | IC50 | = | 105 | nM | ALA4805264 | 6.98 | nM | Homo sapiens | ||
| 9. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | F | = | 73 | % | ALA4805263 | % | ||||
| 10. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | t1/2 | = | 0.74 | hr | ALA4805262 | hr | ||||
| 11. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | Kel | = | 0.94 | /hr | ALA4805261 | /hr | ||||
| 12. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | AUC | = | 1573.33 | ng.hr/ml | ALA4805260 | ng.hr.mL-1 | ||||
| 13. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | Cmax | = | 1161 | ng/ml | ALA4805259 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 14. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | Stabilty | 0 | ALA4805253 | Stable | % | |||||
| 15. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | INH | 0 | ALA4805252 | Active | % | Homo sapiens | ||||
| 16. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | INH | 0 | ALA4805251 | Active | % | Homo sapiens | ||||
| 17. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | IC50 | = | 8765 | nM | ALA4805249 | 5.06 | nM | Homo sapiens | ||
| 18. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | IC50 | = | 65 | nM | ALA4805248 | 7.19 | nM | Homo sapiens | ||
| 19. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | IC50 | = | 35 | nM | ALA4805247 | 7.46 | nM | Homo sapiens | ||
| 20. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | IC50 | = | 36 | nM | ALA4805246 | 7.44 | nM | Homo sapiens |
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