| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5072201 | 25 | Activity | 0 | ALA5035921 | Non-Toxic | ||||||
| 2. | ALA5072201 | 25 | Activity | 0 | ALA5035920 | Non-Toxic | ||||||
| 3. | ALA5072201 | 25 | Drug metabolism | 0 | ALA5035917 | Metabolite_Notdetected | ||||||
| 4. | ALA5072201 | 25 | logD | = | 2.3 | ALA5035909 | ||||||
| 5. | ALA5072201 | 25 | INH | = | 10 | % | ALA5035904 | % | ||||
| 6. | ALA5072201 | 25 | INH | = | 20 | % | ALA5035900 | % | ||||
| 7. | ALA5072201 | 25 | Drug metabolism | 0 | ALA5035899 | Metabolite_Notdetected | ||||||
| 8. | ALA5072201 | 25 | Drug metabolism | 0 | ALA5035898 | Metabolite_Detected | ||||||
| 9. | ALA5072201 | 25 | Drug metabolism | 0 | ALA5035897 | Metabolite_Detected | ||||||
| 10. | ALA5072201 | 25 | t1/2 | > | 55 | min | ALA5035896 | hr | ||||
| 11. | ALA5072201 | 25 | Activity | 0 | ALA5035895 | Non-Toxic | ||||||
| 12. | ALA5072201 | 25 | AUC | = | 962 | microg.hr/mL | ALA5035894 | ng.hr.mL-1 | ||||
| 13. | ALA5072201 | 25 | Activity | = | 57 | % | ALA5035892 | % | Rattus norvegicus | |||
| 14. | ALA5072201 | 25 | IC50 | = | 1.3 | nM | ALA5035891 | 8.89 | nM | |||
| 15. | ALA5072201 | 25 | IC50 | = | 13 | nM | ALA5035890 | 7.89 | nM | |||
| 16. | ALA5072201 | 25 | INH | 0 | ALA5035889 | Dose-Dependent Effect | % | |||||
| 17. | ALA5072201 | 25 | solubility | = | 705 | ug ml-1 | ALA5035885 | ug.mL-1 | ||||
| 18. | ALA5072201 | 25 | solubility | = | 389 | ug ml-1 | ALA5035884 | ug.mL-1 | ||||
| 19. | ALA5072201 | 25 | t1/2 | > | 120 | min | ALA5035883 | hr | ||||
| 20. | ALA5072201 | 25 | t1/2 | > | 120 | min | ALA5035882 | hr |
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