| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5074870 | 7 | F | = | 25 | % | ALA5030430 | % | ||||
| 2. | ALA5074870 | 7 | AUC | = | 5.27 | uM.hr | ALA5030429 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 3. | ALA5074870 | 7 | t1/2 | = | 2.8 | hr | ALA5030428 | hr | ||||
| 4. | ALA5074870 | 7 | Vdss | = | 1.44 | L/Kg | ALA5030427 | L.kg-1 | ||||
| 5. | ALA5074870 | 7 | CL | = | 14.9 | ml/min.kg | ALA5030426 | mL.min-1.kg-1 | ||||
| 6. | ALA5074870 | 7 | t1/2 | = | 1.9 | hr | ALA5030425 | hr | ||||
| 7. | ALA5074870 | 7 | AUClast | = | 5.27 | uM.hr | ALA5030423 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 8. | ALA5074870 | 7 | Cmax | = | 1.11 | uM | ALA5030421 | nM | ||||
| 9. | ALA5074870 | 7 | Cp(f) | = | 36 | nM | ALA5030420 | nM | ||||
| 10. | ALA5074870 | 7 | Activity | 0 | ALA5030419 | Active | ||||||
| 11. | ALA5074870 | 7 | Ki | = | 3.6 | nM | ALA5030418 | 8.44 | nM | Rattus norvegicus | ||
| 12. | ALA5074870 | 7 | Ki | > | 10 | uM | ALA5030417 | nM | Homo sapiens | |||
| 13. | ALA5074870 | 7 | Ki | > | 10 | uM | ALA5030416 | nM | Homo sapiens | |||
| 14. | ALA5074870 | 7 | Ki | = | 3.5 | uM | ALA5030415 | 5.46 | nM | Homo sapiens | ||
| 15. | ALA5074870 | 7 | IC50 | = | 12 | nM | ALA5030414 | 7.92 | nM | Homo sapiens | ||
| 16. | ALA5074870 | 7 | Ki | = | 4 | nM | ALA5030413 | 8.40 | nM | Homo sapiens |
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