| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5075047 | 24 | Drug metabolism | = | 4.1 | % | ALA5044220 | % | ||||
| 2. | ALA5075047 | 24 | Activity | = | 60 | % | ALA5044212 | % | Homo sapiens | |||
| 3. | ALA5075047 | 24 | Activity | 0 | ALA5044210 | Non-Toxic | ||||||
| 4. | ALA5075047 | 24 | Activity | 0 | ALA5044209 | Non-Toxic | ||||||
| 5. | ALA5075047 | 24 | Activity | 0 | ALA5044208 | Non-Toxic | ||||||
| 6. | ALA5075047 | 24 | FC | = | 2.5 | ALA5044207 | ||||||
| 7. | ALA5075047 | 24 | FC | = | 5 | ALA5044206 | ||||||
| 8. | ALA5075047 | 24 | FC | = | 3 | ALA5044205 | ||||||
| 9. | ALA5075047 | 24 | AUC | = | 16 | uM/hr | ALA5044204 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 10. | ALA5075047 | 24 | Activity | 0 | ALA5044203 | Non-Toxic | ||||||
| 11. | ALA5075047 | 24 | Drugexcretion | = | 5 | % | ALA5044202 | % | ||||
| 12. | ALA5075047 | 24 | IC50 | = | 5.7 | uM | ALA5044198 | 5.24 | nM | Homo sapiens | ||
| 13. | ALA5075047 | 24 | MRT | = | 4.8 | hr | ALA5044197 | hr | ||||
| 14. | ALA5075047 | 24 | CL | = | 29 | ml/min.kg | ALA5044196 | mL.min-1.kg-1 | ||||
| 15. | ALA5075047 | 24 | Papp | = | 30 | 10^-6 cm/s | ALA5044195 | 10^-6 cm/s | ||||
| 16. | ALA5075047 | 24 | Therm_solubility | = | 0.03 | mg/ml | ALA5044186 | ug.mL-1 | ||||
| 17. | ALA5075047 | 24 | fIC50 | = | 2.6 | nM | ALA5044165 | nM | Homo sapiens | |||
| 18. | ALA5075047 | 24 | Activity | 0 | ALA5044159 | Non-Toxic | Salmonella enterica subsp. enterica serovar Typhimurium | |||||
| 19. | ALA5075047 | 24 | Activity | 0 | ALA5044158 | Non-Toxic | Salmonella enterica subsp. enterica serovar Typhimurium | |||||
| 20. | ALA5075047 | 24 | Activity | 0 | ALA5044157 | Non-Toxic | Salmonella enterica subsp. enterica serovar Typhimurium |
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