| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5076343 | 24e | Activity | 0 | ALA5032353 | Toxic | ||||||
| 2. | ALA5076343 | 24e | Ki | = | 2.2 | nM | ALA5032352 | 8.66 | nM | Homo sapiens | ||
| 3. | ALA5076343 | 24e | IC50 | > | 10000 | nM | ALA5032351 | nM | Homo sapiens | |||
| 4. | ALA5076343 | 24e | IC50 | = | 80.2 | nM | ALA5032350 | 7.10 | nM | Homo sapiens | ||
| 5. | ALA5076343 | 24e | GI50 | = | 6.2 | uM | ALA5032349 | nM | Mus musculus | |||
| 6. | ALA5076343 | 24e | GI50 | = | 6.1 | uM | ALA5032348 | nM | Mus musculus | |||
| 7. | ALA5076343 | 24e | Kel | = | 0.355 | /hr | ALA5032347 | /hr | ||||
| 8. | ALA5076343 | 24e | t1/2 | = | 1.97 | hr | ALA5032346 | hr | ||||
| 9. | ALA5076343 | 24e | Tmax | = | 0.25 | hr | ALA5032345 | hr | ||||
| 10. | ALA5076343 | 24e | C0 | 0 | ALA5032344 | Not Determined | ||||||
| 11. | ALA5076343 | 24e | Cmax | = | 1586 | ng/ml | ALA5032343 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 12. | ALA5076343 | 24e | AUCt | = | 1766 | hr.ng/ml | ALA5032342 | ng.hr.mL-1 | ||||
| 13. | ALA5076343 | 24e | AUC | = | 1808 | hr.ng/ml | ALA5032341 | ng.hr.mL-1 | ||||
| 14. | ALA5076343 | 24e | CL | 0 | ALA5032340 | Not Determined | ||||||
| 15. | ALA5076343 | 24e | Vd | 0 | ALA5032339 | Not Determined | ||||||
| 16. | ALA5076343 | 24e | MRT | = | 1.41 | hr | ALA5032338 | hr | ||||
| 17. | ALA5076343 | 24e | F | = | 30.3 | % | ALA5032337 | % | ||||
| 18. | ALA5076343 | 24e | Kel | = | 0.497 | /hr | ALA5032336 | /hr | ||||
| 19. | ALA5076343 | 24e | t1/2 | = | 1.89 | hr | ALA5032335 | hr | ||||
| 20. | ALA5076343 | 24e | Cmax | = | 2160 | ng/ml | ALA5032334 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM |
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