# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5078027 | [64Cu]Cu-NODAGA-TATE | SUV | = | 0.08 | ALA5043881 | ||||||
2. | ALA5078027 | [64Cu]Cu-NODAGA-TATE | SUVmax | = | 3 | ALA5043875 | ||||||
3. | ALA5078027 | [64Cu]Cu-NODAGA-TATE | Drug uptake | = | 15 | % | ALA5043873 | % | ||||
4. | ALA5078027 | [64Cu]Cu-NODAGA-TATE | SUV | = | 2.4 | ALA5043872 | ||||||
5. | ALA5078027 | [64Cu]Cu-NODAGA-TATE | Drug uptake | = | 9.5 | ALA5043871 | ||||||
6. | ALA5078027 | [64Cu]Cu-NODAGA-TATE | Drug uptake | = | 45 | % | ALA5043870 | % | ||||
7. | ALA5078027 | [64Cu]Cu-NODAGA-TATE | t1/2 | 0 | ALA5043869 | Not Determined | ||||||
8. | ALA5078027 | [64Cu]Cu-NODAGA-TATE | t1/2 | > | 24 | hr | ALA5043868 | hr | ||||
9. | ALA5078027 | [64Cu]Cu-NODAGA-TATE | Bmax | = | 383 | fmol/mg | ALA5043867 | fmol/mg | Mus musculus | |||
10. | ALA5078027 | [64Cu]Cu-NODAGA-TATE | Kd | = | 2.89 | nM | ALA5043866 | 8.54 | nM | Mus musculus | ||
11. | ALA5078027 | [64Cu]Cu-NODAGA-TATE | Kd | > | 300 | uM | ALA5043865 | nM | Homo sapiens | |||
12. | ALA5078027 | [64Cu]Cu-NODAGA-TATE | logD | = | -3.43 | ALA5043864 | ||||||
13. | ALA5078027 | [64Cu]Cu-NODAGA-TATE | PB | < | 30 | % | ALA5043863 | % | Homo sapiens | |||
14. | ALA5078027 | [64Cu]Cu-NODAGA-TATE | PPB | = | 46 | % | ALA5043862 | % |