# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5081275 | 6 | INH | = | 10 | % | ALA5034372 | % | Homo sapiens | |||
2. | ALA5081275 | 6 | INH | = | 10 | % | ALA5034371 | % | ||||
3. | ALA5081275 | 6 | deltaT | = | 1.7 | degrees C | ALA5034370 | degrees C | Homo sapiens | |||
4. | ALA5081275 | 6 | Drug uptake | 0 | ALA5034369 | Active | ||||||
5. | ALA5081275 | 6 | INH | 0 | ALA5034368 | Not Active | % | Homo sapiens | ||||
6. | ALA5081275 | 6 | INH | 0 | ALA5034367 | Not Active | % | Homo sapiens | ||||
7. | ALA5081275 | 6 | INH | 0 | ALA5034366 | Not Active | % | |||||
8. | ALA5081275 | 6 | Selectivity ratio | = | 1000 | ALA5034365 | ||||||
9. | ALA5081275 | 6 | Selectivity ratio | = | 1000 | ALA5034364 | ||||||
10. | ALA5081275 | 6 | Selectivity ratio | = | 10000 | ALA5034363 | ||||||
11. | ALA5081275 | 6 | Selectivity ratio | = | 10000 | ALA5034362 | ||||||
12. | ALA5081275 | 6 | Selectivity ratio | = | 10000 | ALA5034361 | ||||||
13. | ALA5081275 | 6 | Selectivity ratio | = | 10000 | ALA5034360 | ||||||
14. | ALA5081275 | 6 | INH | 0 | ALA5034359 | Not Active | % | |||||
15. | ALA5081275 | 6 | Km | = | 0.16 | nM | ALA5034358 | nM | Homo sapiens | |||
16. | ALA5081275 | 6 | Km | = | 0.64 | nM | ALA5034357 | nM | Homo sapiens | |||
17. | ALA5081275 | 6 | Ki | = | 0.61 | nM | ALA5034356 | 9.21 | nM | Homo sapiens | ||
18. | ALA5081275 | 6 | alphaKi | = | 2.1 | nM | ALA5034355 | nM | Homo sapiens | |||
19. | ALA5081275 | 6 | Ki(app) | = | 1 | nM | ALA5034354 | 9.00 | nM | Homo sapiens | ||
20. | ALA5081275 | 6 | IC50 | = | 4.1 | nM | ALA5034353 | 8.39 | nM | Homo sapiens |